Triptorelin (GNRH ) 100mcg
- The empirical formula is C64H82N18O13 • C23H16O6
- Molecular weight is 1699.9
Triptorelin Restores Bodybuilder’s Hormones
If you are a bodybuilder, then chances are that you will have to take some form of hormone replacement therapy (HRT) at some point in your career. One of the most popular hormones used for this purpose is triptorelin, which is a synthetic version of the luteinizing hormone-releasing hormone (LHRH).
LHRH is responsible for stimulating the production of testosterone and other hormones in the body. Triptorelin works by mimicking the action of LHRH, which allows it to stimulate the production of testosterone and other hormones.
What is Triptorelin?
Triptorelin is a synthetic decapeptide analogue of gonadotropin-releasing hormone (GnRH). It belongs to a class of drugs called gonadotropin-releasing hormone agonists. By acting on the pituitary gland, these drugs decrease the production of testosterone, estrogen, and other sex hormones in the body.
Triptorelin was originally developed to treat prostate cancer in men. But it is now more commonly used for other medical applications like treating precocious puberty, endometriosis, uterine fibroids, and as part of in-vitro fertilization protocols.
For bodybuilders and athletes, triptorelin is used to dramatically reduce endogenous testosterone and estrogen production. This induces a temporary chemical castration state, allowing for effective post-cycle therapy following a steroid cycle.
What are the Benefits of Using Triptorelin?
Here are some of the key benefits bodybuilders look for when using triptorelin as part of their post-cycle therapy:
- It rapidly lowers testosterone levels to help recover natural hormone function after a steroid cycle
- Reduces estrogen conversion from aromatization to mitigate estrogenic side effects
- It avoids testosterone suppression or renal toxicity issues seen with SERMs like nolvadex
- More thoroughly restores the HPTA axis compared to selective estrogen receptor modulators
- Induces greater release of luteinizing hormone and follicle-stimulating hormone to stimulate testosterone production
- Short 2-3-week dosing makes it convenient for short PCT periods
- Enables faster clearance of any remaining exogenous steroids still circulating post-cycle
Overall, triptorelin is a highly effective medication for hormonal recovery after suppressive androgenic steroid cycles. The temporary induced hypogonadism allows the body to upregulate receptors and resume natural testosterone production quickly after discontinuing use.
How to Take Triptorelin for Best Results
Here are some guidelines on using triptorelin for successful post-cycle therapy:
- Standard dosing is 2-3 injections of 100 mcg per injection, spaced 1 week apart
- The first injection should be given around 2 weeks after last steroid dose or when exogenous steroid levels are declining
- Follow with a second 100-mcg injection 7 days after the first
- Optionally, administer a third 100-mcg dose 7 days after the second injection
- 2 injections is sufficient for lighter cycles; 3 doses provides maximum HPTA suppression for heavier cycles
- Always use sterile technique and inject subcutaneously into fat layer of lower abdominal area
- Discontinue use once post-cycle therapy is complete
Following this protocol, triptorelin stimulates maximum natural testosterone production to restore pre-cycle hormone balance in a short timeframe.
Potential Side Effects of Triptorelin
While generally well tolerated, potential triptorelin side effects should be considered:
- Temporary testosterone suppression – This is the intent, but results in fatigue, low libido, erectile dysfunction and other hypogonadism symptoms during use
- Estrogen rebound – Estrogen may spike after ending triptorelin before testosterone levels recover
- Increased risk of depression, anxiety, and irritability – Low hormone levels can impact mental health
- Headache, dizziness, nausea – Transient side effects may occur after injecting
- Hot flashes and night sweats – Users may experience “menopausal” symptoms from low-sex hormones
- Reduction in bone mineral density – Lack of sex hormones decreases bone mass
However, side effects resolve within 1-2 months after stopping use as normal hormonal balance is restored. Using aromatase inhibitors and hormone testing helps mitigate side effects during recovery.
How to Minimize Triptorelin Side Effects
Here are some strategies to help reduce potential side effects:
- Follow sensible dosing protocols – Use the minimum effective doses and duration
- Use aromatase inhibitors like exemestane to prevent estrogen rebound
- Get bloodwork to confirm hormone levels are recovering properly
- Include hCG during the last 2 weeks of the cycle to prime natural testosterone function
- Implement on-cycle supplements like DHEA to support hormone balance
- Adopt healthy lifestyle habits – train, eat well and sleep enough to aid recovery
- Time-on-cycle steroid use appropriately and allow sufficient time off between cycles
- Monitor mental health and get medical assistance if depression or anxiety develops
With careful use limited to occasional PCT, healthy men can safely use triptorelin for post-cycle therapy.
What is the Best Triptorelin Dosage and Timing?
For optimal results, adhere to the following triptorelin dosage guidelines:
- Dosage: 100 mcg administered subcutaneously
- Injection frequency: Every 7 days
- Total doses: 2-3 injections (200–300 mg total)
Start administering triptorelin about 2 weeks after your last steroid dose. This ensures exogenous hormone levels are declining before inducing suppression.
Use a dosage of 100 mcg and repeat the same dosage every 7 days. Two 100 mcg doses 1 week apart (200 mcg total) is often sufficient for lighter steroid cycles.
For heavy or longer steroid cycles, a third 100 mcg injection may be warranted to ensure full HPTA suppression. This provides more comprehensive PCT support.
Always follow sterile injection procedures. Rotate injection sites to avoid irritation. Discontinue use once post-cycle therapy is complete.
Where Can I Buy Triptorelin Online?
There are a few possible sources to purchase triptorelin online:
- Medical clinics – Legitimate anti-aging or men’s health clinics may prescribe triptorelin for hormone optimization purposes
- Overseas pharmacies – Some foreign online pharmacies loosely dispense triptorelin, but product quality and legality may be questionable
- Peptide companies – A handful of research peptide companies offer triptorelin for research purposes only
- Underground labs – Bodybuilding forums and networks may provide access to lab-made triptorelin from underground sources
However, accessibility has become more limited in recent years due to increased regulation of these drugs. Pharmaceutical-grade triptorelin can still be obtained through proper medical channels or specialty anti-aging clinics. But always exercise caution when purchasing any prescription drug online.
In summary, when used properly Triptorelin is a highly effective medical treatment for hormonal recovery after suppressive anabolic steroid usage. It reliably restores the HPTA axis to bring testosterone and estrogen back to normal physiological ranges. But it should be treated with care and respect, like Buypeptidesusa, a clinical pharmacy-grade medication.